Stereospecific Synthesis of 2,3-Dimethoxy-naphtho[1,2-b]indolizidine
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منابع مشابه
Stereospecific synthesis of amphetamines
Regioselective addition of aryl lithium to commercially available (S)-(+)-propylene oxide provides the corresponding (S)-aryl-2-propanol. The (R)-amphetamine is obtained by conversion of the alcohol to the tosylate followed by azide displacement and hydrogenation. Mitsunobu conversion of the alcohol to the (R)-bromide followed by azide displacement and hydrogenation affords the (S)-amphetamine....
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ژورنال
عنوان ژورنال: Archiv der Pharmazie
سال: 1989
ISSN: 0365-6233,1521-4184
DOI: 10.1002/ardp.19893221008